Formestane -
• Formestane increases IGF-1 secretion and activity.
• Formestane decreases the number of progesterone receptors (inhibits the trenbolone and “deca-dick” type side effects and increases fat loss)
• Formestane inhibits 91.9% of aromatase enzyme production
• Formestane increases HPTA activity similar to HCG and Clomid together
• Formestane is anabolic and androgenic
• Formestane is a “suicide inhibitor” of aromatase. Formestane decreases SHBG 34% thus increasing androgen activity.
• Formestane inhibits DHT (dehydrotestosterone) formation and activity.
• Formestane possesses 1% of the binding affinity of DHT to DHT receptors
• Formestane has been shown to decrease prostate concerns such as BPH.
• Formestane has been shown to continue to increase HPTA function above natural levels even after 22 weeks of continuous administration
Try cutting the pills into pieces. Most AI's are extremely overdosed imo when it comes to estro control for male lifters on cycle. 6.25mg Aromasin or 0.25mg Arimidex is all most should need for a single dose split up a few times a week at most. That is if we're talking pharm grade that's correctly dosed.
You weren't very clear in your post. Why are you using the aromatase inhibitor? To prevent estro rebound? Will you be on t.r.t?
If your not on H.R.T then a quality over the counter anti estrogen may suffice. If your on a dose of test, even low dose, you may need one of the stronger a.i's such as Exemestane. Aromasin works well for me, a-dex never seemed to work and letro has horrendous sides. Aromasin was effective without any nothing noticeable sides (or at least nothing prolific). I also suffer from estrogen rebound(symptoms that were manageable will just comeback spontaneously when I'm off cycle) so I will be running 6.25 mg per day of exemestane
Continuously. I haven't yet ran it yr round but I'm not expecting any sexual dysfunction etc as far as neg sides.
I hope to give resveratrol (fingers crossed for budget allowing it) a try for a healthy alternative to managing estro symptoms. LK3 has been very helpful in answering any questions I had.
doc advised me 10mg of aromasin per day, has had no adverse side effects at all on my libido , keep in mind i do take 25mg proviron per day during cruise periods also. I am very estrogen sensitive and this does the trick, keep in mind high levels of estrogen don't just cause gyno (which most people seem to use as measure if their estrogen sensitive) it causes a whole host of other problems to.
You should definitely split up the doses. It's very effective. If you're taking the recommended 100-150 mgs. a day then add a few mgs. of copper and you'll be good to go.
You should definitely split up the doses. It's very effective. If you're taking the recommended 100-150 mgs. a day then add a few mgs. of copper and you'll be good to go.