Steroid Binding Constants

[sbc5966]

Hey All,

Could anybody point me toward a source/table that is a concise reference to steroids and their association constant with the androgen receptor?

I suppose relative binding affinity would be ok, but a true Kd would be sweet.

Even more Kudos if it is split up by tissue type?


Thanks a mil in advance.

 

[andrew.peplin]

I'm interested in an article on this also.

 

[bomb401]

Just find the androgenic/anabolic ratios...

 

[collinb]

Found this on a forum, androgenic to anabolic ratios!




Compound:----------------------------------------------Androgenic------Anabolic
1-Testosterone--------------------------------------------100----------------200
Anabolicum Vister(Quinbolone)(oral Boldenone)----50------100
Anadrol 50(Oxymetholone)------------------------------45------320
Anadur(Nandrolone Hexyloxyphenylpropionate)----37-----125
Anatrofin(Stenbolone Acetate)-------------------------107-144-----267-332
Anavar(Oxandrolone)-------------------------------------24------322-630
Andractim(Dihydrotestosteron)-------------------------30-260-----60-220
Andriol(Testosterone Undecanoate)------------------100------100
Androderm(Testosterone)------------------------------100------100
Androgel(Testosterone)---------------------------------100------100
Boldabol(Boldenone Acetate)---------------------------50------100
Cheque Drops(Mibolerone)-----------------------------1,800------4,100
Danocrine(Danazol)---------------------------------------37------125
Deca-Durabolin(Nandrolone Decanoate)--------------37------125
Deposterona(Testosterone Blend)---------------------100------100
Dianabol(Methandrostenolone)----------------------40-60------90-210
Dimethyltrienolone-------------------------------------10,000+-----10,000+
Dinandrol(Nandrolone Blend)---------------------------37------125
Durabolin(NPP)--------------------------------------------37------125
Dynabol(Nandrolone Cypionate)----------------------37------125
Equipoise(Boldenone Undecylenate)-----------------50------100
Esiclene(Formebolone)-----------------------------------No Data Available
Genabol(Norbolethone)--------------------------------17------350
Halotestin(Fluoxymesterone)-------------------------850------1,900
Hydroxytestosterone-----------------------------------25------65
Laurabolin(Nandrolone Laurate)-----------------------37------125
Madol(Desoxymethyltestosterone )------------------187------1,200
Masteron(Drostanolone Propionate)------------------25-40------62-130
Megagrisevit-Mono(Clostebol Acetate)-------------25------46
MENT(Methylnortestosterone Acetate)---------------650------2,300
Mestanolone---------------------------------------------78-254------107
Methandriol(Mythelandrostenedi ol)----------------30-60------20-60
Methyl-1-Testosterone-------------------------------100-220------910-1,600
Methyldienolone----------------------------------------200-300------1,000
Methylhydroxynandrolone(MHN)------------------281------1304
Methyltestosterone---------------------------------94-130------115-150
Metribolone(Methyltrienolone)------------6,000-7,000------12,000-30,000
Miotolan(Furazabol)-------------------------------------73-94------270-330
Myagen(Bolasterone)----------------------------------300------575
Nilevar(Norethandrolone)------------------------------22-55------100-200
Omnadren(Testosterone Blend)-----------------------100------100
Orabolin(Ethylestrenol)---------------------------20-400------200-400
Oral Turinabol--------------------------------------None------100+
Oranabol(Oxymesterone)--------------------------------------50------330
Orgasteron(Normethandrolone)-----------------------325-580------110-125
Parabolan(Tren Hexahydrobenzycarbonate)------------500------500
Primobolan(Methenolone Acetate)---------------------44-57------88
Primobolan Depot(Methenolone Enanthate)----------44-57------88
Prostanozol-------------------------------------------------n/a------n/a
Protabol(Thiomesterone)----------------------------------61------456
Proviron(Mesterolone)----------------------------------------30-40------100-150
Sanabolicum(Nandrolone Cyclohexylpropionate)-------37------125
Steranabol Ritardo(Oxabolone Cypionate)-----------20-60------50-90
Superdrol(Methyldrostanolone)-------------------------400------20
Sustanon 100 & 250---------------------------------------100------100
Synovex(Testosterone Propionate & Estradiol)--------100------100
Test 400-----------------------------------------------------100------100
Test Enanthate/Cyp/Prop/Susp & Blends------------100------100
THG(Tetrahydrogestrinone)-------------------------No Data Available
Tren Acetate/Enanthate & Blends------------------500------500
Winstrol(Stanozolol)------------------------------------30------320

 

[E.J.]

Where do I find some dimethyltrienolone?